Description
SR-9011 is a synthetic REV-ERB agonist, designed to selectively bind and modulate the REV-ERBα and REV-ERBβ nuclear receptors. It plays a role in circadian rhythm regulation, metabolic pathways, and transcriptional control by influencing gene expression linked to lipid and glucose metabolism.
This compound undergoes hepatic metabolism via oxidation and conjugation, with clearance primarily occurring through renal and biliary excretion.